Compile Data Set for Download or QSAR

Found 32 hits of Enzyme Inhibition Constant Data   

TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200547(CHEMBL3949842)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200556(CHEMBL3904435)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200544(CHEMBL3970645)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200545(CHEMBL3965572)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200543(CHEMBL3941088)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200549(CHEMBL3932441)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200550(CHEMBL3905486)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200552(CHEMBL3898411)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200548(CHEMBL3895496)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200551(CHEMBL3978901)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200553(CHEMBL3898379)copy SMILEScopy InChI
Affinity DataKi:  81nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200555(CHEMBL3984293)copy SMILEScopy InChI
Affinity DataKi:  99nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200546(CHEMBL3939229)copy SMILEScopy InChI
Affinity DataKi:  111nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200554(CHEMBL3968765)copy SMILEScopy InChI
Affinity DataKi:  135nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM166683(U74389G (B9))copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200547(CHEMBL3949842)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200556(CHEMBL3904435)copy SMILEScopy InChI
Affinity DataIC50: 105nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200544(CHEMBL3970645)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200545(CHEMBL3965572)copy SMILEScopy InChI
Affinity DataIC50: 146nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200543(CHEMBL3941088)copy SMILEScopy InChI
Affinity DataIC50: 149nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200548(CHEMBL3895496)copy SMILEScopy InChI
Affinity DataIC50: 155nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 45 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200549(CHEMBL3932441)copy SMILEScopy InChI
Affinity DataIC50: 178nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200550(CHEMBL3905486)copy SMILEScopy InChI
Affinity DataIC50: 205nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200552(CHEMBL3898411)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200551(CHEMBL3978901)copy SMILEScopy InChI
Affinity DataIC50: 254nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200548(CHEMBL3895496)copy SMILEScopy InChI
Affinity DataIC50: 254nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200553(CHEMBL3898379)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200555(CHEMBL3984293)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200546(CHEMBL3939229)copy SMILEScopy InChI
Affinity DataIC50: 482nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200554(CHEMBL3968765)copy SMILEScopy InChI
Affinity DataIC50: 586nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM166683(U74389G (B9))copy SMILEScopy InChI
Affinity DataIC50: 910nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
TargetCaspase-5(Homo sapiens (Human))
DePaul University

Curated by ChEMBL
LigandPNGBDBM50200548(CHEMBL3895496)copy SMILEScopy InChI
Affinity DataIC50: 2.56E+3nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 15 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89M0PubMed
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