Found 28 hits of Enzyme Inhibition Constant Data
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 88nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 93nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 982nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 6.60E+3nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: >1.30E+4nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 4.00E+6nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 8.90E+6nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Bristol-Myers Squibb R&D
Curated by ChEMBL
Bristol-Myers Squibb R&D
Curated by ChEMBL
Affinity DataKi: 4.90E+7nMAssay Description:Inhibition of recombinant human factor-7a/TF using S2288 as substrate measured after 60 minsMore data for this Ligand-Target Pair