Compile Data Set for Download or QSAR

Found 17 hits of Enzyme Inhibition Constant Data   

TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142607(CHEMBL3759390)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142603(CHEMBL3759469)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142605(CHEMBL3759527)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142612(CHEMBL3758318)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142606(CHEMBL3758252)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142609(CHEMBL3759138)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142610(CHEMBL3759124)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142608(CHEMBL3759809)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142604(CHEMBL3759334)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142616(CHEMBL3759154)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142611(CHEMBL3759856)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142613(CHEMBL3758779)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50304101((RS)-2-Amino-3-(5,6-dichloro-3'-hydroxybiphenyl-3-...)copy SMILEScopy InChI
Affinity DataKi:  9.23E+4nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142615(CHEMBL3759684)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142614(CHEMBL3758336)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142617(CHEMBL3758644)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50142618(CHEMBL3759959)copy SMILEScopy InChI
Affinity DataKi:  1.05E+5nMAssay Description:Displacement of [3H]SYM2081 from recombinant rat GluK1(Q)1b receptor expressed in sf9 cells incubated for 1 to 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34JKPubMed
* indicates data uncertainty>20%