Compile Data Set for Download or QSAR

Found 8 hits of Enzyme Inhibition Constant Data   

TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116040((7-{3-[3-(4-Nitro-phenyl)-ureidomethyl]-pyrrol-1-y...)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116044(CHEMBL416685 | {6-Nitro-2,3-dioxo-7-[3-(4-phenyl-p...)copy SMILEScopy InChI
Affinity DataKi:  530nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116042(CHEMBL63861 | {7-[3-(4-Benzyl-piperazin-1-ylmethyl...)copy SMILEScopy InChI
Affinity DataKi:  680nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116048(CHEMBL67828 | {6-Nitro-2,3-dioxo-7-[3-(4-phenethyl...)copy SMILEScopy InChI
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116047((6-Nitro-2,3-dioxo-7-{3-[(3-phenyl-propylamino)-me...)copy SMILEScopy InChI
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116043(3-(6-Nitro-2,3-dioxo-7-pyrrol-1-yl-3,4-dihydro-2H-...)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116050(1-(4-Carboxymethyl-7-nitro-2,3-dioxo-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  4.10E+3nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Abbott GmbH & Co. KG

Curated by ChEMBL
LigandPNGBDBM50116041(CHEMBL303415 | [6-Nitro-2,3-dioxo-7-(3-piperidin-1...)copy SMILEScopy InChI
Affinity DataKi:  5.70E+3nMAssay Description:Binding affinity towards cloned human GluR7 subunit stably expressed in cultured HEK-293 cells using [3]H-kainate as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22806XKPubMed
* indicates data uncertainty>20%