Compile Data Set for Download or QSAR

Found 2 hits of Enzyme Inhibition Constant Data   

TargetHistone deacetylase 1(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)

Curated by ChEMBL
LigandPNGBDBM50503690(CHEMBL4456445)copy SMILEScopy InChI
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of human full length C-terminal FLAG/His-tagged HDAC1 expressed in baculovirus infected Sf9 insect cells using Lys-Ac-AMC as substrate mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44TJZPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)

Curated by ChEMBL
LigandPNGBDBM50503692(CHEMBL4437833)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length C-terminal FLAG/His-tagged HDAC1 expressed in baculovirus infected Sf9 insect cells using Lys-Ac-AMC as substrate mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44TJZPubMed
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