Found 4 hits of Enzyme Inhibition Constant Data
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair
TargetHistone deacetylase 5(Homo sapiens (Human))
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Charles River Discovery (previously BioFocus)
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human C-terminal His-tagged HDAC5 catalytic domain (656 to 1122 residues) expressed in baculovirus infected Sf9 insect cells using Boc-...More data for this Ligand-Target Pair