Compile Data Set for Download or QSAR

Found 14 hits of Enzyme Inhibition Constant Data   

TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50467705(CHEMBL4282830)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519492(CHEMBL1233663)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Inhibition of human HGPRT assessed as inhibitor constant for enzyme-inhibitor-substrate complex formation using [5'-14C]IMP as substrate by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50467710(CHEMBL4290716)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519500(CHEMBL1233603)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Inhibition of human HGPRT assessed as inhibitor constant for enzyme-inhibitor-substrate complex formation using [5'-14C]IMP as substrate by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519500(CHEMBL1233603)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Inhibition of human HGPRT assessed as inhibitor constant for enzyme-inhibitor complex formation using [5'-14C]IMP as substrate by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519497(CHEMBL4546337)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519492(CHEMBL1233663)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Inhibition of human HGPRT assessed as inhibitor constant for enzyme-inhibitor complex formation using [5'-14C]IMP as substrate by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519504(CHEMBL4561412)copy SMILEScopy InChI
Affinity DataKi:  400nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519501(CHEMBL4583093)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Inhibition of human N-terminal His6-tagged HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519505(CHEMBL4578350)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human N-terminal His6-tagged HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519493(CHEMBL4453040)copy SMILEScopy InChI
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519502(CHEMBL4452934)copy SMILEScopy InChI
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human N-terminal His6-tagged HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519496(CHEMBL4439813)copy SMILEScopy InChI
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50519503(CHEMBL2420976)copy SMILEScopy InChI
Affinity DataKi:  7.30E+7nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by Hanes-plot based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1571NPubMed
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