Found 32 hits of Enzyme Inhibition Constant Data
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in HEK293 cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Antagonist activity at human MT2 receptorMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 87nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 91nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 167nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 246nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Binding affinity to MT2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) assessed as cAMP accumulationMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University in Cairo
Curated by ChEMBL
The German University in Cairo
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) assessed as cAMP accumulationMore data for this Ligand-Target Pair