Compile Data Set for Download or QSAR

Found 5 hits of Enzyme Inhibition Constant Data   

TargetNeuromedin-U receptor 2(Mus musculus)
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049425(CHEMBL3356083)copy SMILEScopy InChI
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse NMUR2 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049422(CHEMBL3315335)copy SMILEScopy InChI
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049423(CHEMBL3315278)copy SMILEScopy InChI
Affinity DataEC50:  8.40nMAssay Description:Partial agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
TargetNeuromedin-U receptor 2(Mus musculus)
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049426(CHEMBL3356082)copy SMILEScopy InChI
Affinity DataEC50:  156nMAssay Description:Agonist activity at mouse NMUR2 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University of Pharmacy and Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)copy SMILEScopy InChI
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z71PubMed
* indicates data uncertainty>20%