Found 35 hits of Enzyme Inhibition Constant Data
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.65nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.04E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.07E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.78E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 2.04E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 2.62E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 3.51E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 3.94E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 4.98E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 5.03E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 6.98E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 7.12E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 7.22E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 9.88E+3nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of L-[3H]Nicotine from alpha4beta2 nAChR in rat brain homogenate by rapid filtration methodMore data for this Ligand-Target Pair
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