Compile Data Set for Download or QSAR

Found 1 hit of Enzyme Inhibition Constant Data   

TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Chugai Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM206104(US9255110, 17)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged RAF1 catalytic domain (306 to 648 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6F3RPubMed
* indicates data uncertainty>20%