Found 5 hits of Enzyme Inhibition Constant Data
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University of Vienna
Curated by ChEMBL
Medical University of Vienna
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]WIN35428 from human DAT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University of Vienna
Curated by ChEMBL
Medical University of Vienna
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]WIN35428 from human DAT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University of Vienna
Curated by ChEMBL
Medical University of Vienna
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity to DAT (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University of Vienna
Curated by ChEMBL
Medical University of Vienna
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to DAT (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Medical University of Vienna
Curated by ChEMBL
Medical University of Vienna
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]WIN35428 from human DAT after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair