Found 22 hits of Enzyme Inhibition Constant Data
Affinity DataEC50: 10nMAssay Description:Efficacy against phenylephrine precontracted tissue relaxation in rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 560nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2B receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2B receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 97nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 950nMAssay Description:Relative efficacy against phenylephrine precontracted tissue relaxation in Guinea pig aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 6.70nMAssay Description:Efficacy against phenylephrine precontracted tissue relaxation in rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Efficacy against phenylephrine precontracted tissue relaxation in rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Efficacy against phenylephrine precontracted tissue relaxation in rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 8.80nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2B receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.14E+3nMAssay Description:Relative efficacy against phenylephrine precontracted tissue relaxation in Guinea pig aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Relative efficacy against phenylephrine precontracted tissue relaxation in Guinea pig aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 680nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2B receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2B receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 440nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2B receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2B receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Relative efficacy against phenylephrine precontracted tissue relaxation in Guinea pig aortaMore data for this Ligand-Target Pair