Found 6 hits of Enzyme Inhibition Constant Data
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataEC50: 1.40nMAssay Description:Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by rapid filtration ass...More data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataEC50: 1.14E+3nMAssay Description:Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by rapid filtration ass...More data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataEC50: 0.0360nMAssay Description:Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by rapid filtration ass...More data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by rapid filtration ass...More data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataEC50: 945nMAssay Description:Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by rapid filtration ass...More data for this Ligand-Target Pair
TargetUracil nucleotide/cysteinyl leukotriene receptor(Homo sapiens (Human))
University of Pavia
Curated by ChEMBL
University of Pavia
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by rapid filtration ass...More data for this Ligand-Target Pair