Compile Data Set for Download or QSAR

Found 35 hits of Enzyme Inhibition Constant Data   

TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50147093(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of human kidney uPA using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of human kidney uPA using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of human kidney uPA using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human kidney uPA using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetProthrombin(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasminogen(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of plasmin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetTrypsin(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of trypsin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetTrypsin(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of trypsin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetProthrombin(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasminogen(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of plasmin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of human plasma kallikrein using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of human plasma kallikrein using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetProthrombin(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasminogen(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of plasmin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasminogen(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of plasmin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of tPA (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of tPA (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetProthrombin(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of activated protein C (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of activated protein C (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor X(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of factor 10a (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human plasma kallikrein using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor X(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of factor 10a (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human plasma kallikrein using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of activated protein C (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of activated protein C (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor X(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50459055(CHEMBL4207715)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of factor 10a (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor X(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of factor 10a (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
University of Wollongong

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
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