Found 16 hits of Enzyme Inhibition Constant Data
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 334nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze
Curated by ChEMBL
Universit£ degli Studi di Firenze
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
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