Compile Data Set for Download or QSAR

Found 16 hits of Enzyme Inhibition Constant Data   

TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545314(CHEMBL4643397)copy SMILEScopy InChI
Affinity DataIC50: 0.340nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545312(CHEMBL4632532)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545311(CHEMBL4643898)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545312(CHEMBL4632532)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545313(CHEMBL4644153)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545316(CHEMBL4633630)copy SMILEScopy InChI
Affinity DataIC50: 146nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545317(CHEMBL4645283)copy SMILEScopy InChI
Affinity DataIC50: 156nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545322(CHEMBL4642713)copy SMILEScopy InChI
Affinity DataIC50: 334nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545318(CHEMBL4647074)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545314(CHEMBL4643397)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545315(CHEMBL4646158)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545322(CHEMBL4642713)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545321(CHEMBL4634083)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545320(CHEMBL4632626)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545319(CHEMBL4646403)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£ degli Studi di Firenze

Curated by ChEMBL
LigandPNGBDBM50545313(CHEMBL4644153)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3BFSPubMed
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