Compile Data Set for Download or QSAR

Found 19 hits of Enzyme Inhibition Constant Data   

TargetD(3) dopamine receptor(Homo sapiens (Human))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382290(CARIPRAZINE HYDROCHLORIDE | RGH-188 HCL)copy SMILEScopy InChI
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to human dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382312(CHEMBL2024677)copy SMILEScopy InChI
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382310(CHEMBL2024675)copy SMILEScopy InChI
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382290(CARIPRAZINE HYDROCHLORIDE | RGH-188 HCL)copy SMILEScopy InChI
Affinity DataKi:  0.810nMAssay Description:Binding affinity to human dopamine D2S receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMedDrugBank
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382306(CHEMBL2024522)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382311(CHEMBL2024676)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382307(CHEMBL2024523)copy SMILEScopy InChI
Affinity DataKi:  4.95nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382309(CHEMBL2024525)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382290(CARIPRAZINE HYDROCHLORIDE | RGH-188 HCL)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Binding affinity to human dopamine D2L receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMedDrugBank
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382310(CHEMBL2024675)copy SMILEScopy InChI
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382308(CHEMBL2024524)copy SMILEScopy InChI
Affinity DataKi:  13.1nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382305(CHEMBL2024521)copy SMILEScopy InChI
Affinity DataKi:  15.9nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382306(CHEMBL2024522)copy SMILEScopy InChI
Affinity DataKi:  19.8nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382312(CHEMBL2024677)copy SMILEScopy InChI
Affinity DataKi:  20.2nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382307(CHEMBL2024523)copy SMILEScopy InChI
Affinity DataKi:  53.4nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382305(CHEMBL2024521)copy SMILEScopy InChI
Affinity DataKi:  94nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382309(CHEMBL2024525)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382311(CHEMBL2024676)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50382308(CHEMBL2024524)copy SMILEScopy InChI
Affinity DataKi:  392nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1MZNPubMed
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