Found 11 hits of Enzyme Inhibition Constant Data
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 413nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Affinity to NK3 receptors assayed by displacement of [125I]-Bolton-Hunter labeled eledoisin radioligandMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to the NK2 receptor assayed by displacement of [125I]-Neurokinin AMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards cloned neurokinin 1 receptor, based on the displacement of [125I]-labeled substance PMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Rattus norvegicus (rat))
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Merck, Sharp and Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.92E+5nMAssay Description:The inhibitory concentration of the compound against rat neurokinin-1 receptorMore data for this Ligand-Target Pair
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