Found 6 hits of Enzyme Inhibition Constant Data
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 2.38nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 97.7nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 893nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 1.71E+3nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 3.62E+3nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair