Compile Data Set for Download or QSAR

Found 5 hits of Enzyme Inhibition Constant Data   

TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Novartis Pharma Research

Curated by ChEMBL
LigandPNGBDBM50097954(7-Cyclopentyl-5-(4-methoxy-phenyl)-7H-pyrrolo[2,3-...)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of v-Abl tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3RMFPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Novartis Pharma Research

Curated by ChEMBL
LigandPNGBDBM50088900(5,7-Diphenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine ...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of p60 c-Src tyrosine kinase enzymeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3RMFPubMed
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Novartis Pharma Research

Curated by ChEMBL
LigandPNGBDBM50097954(7-Cyclopentyl-5-(4-methoxy-phenyl)-7H-pyrrolo[2,3-...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of v-Abl tyrosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3RMFPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Novartis Pharma Research

Curated by ChEMBL
LigandPNGBDBM50097954(7-Cyclopentyl-5-(4-methoxy-phenyl)-7H-pyrrolo[2,3-...)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of Epidermal growth factor receptor (EGF-R) tyrosine kinase activity More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3RMFPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Novartis Pharma Research

Curated by ChEMBL
LigandPNGBDBM50097954(7-Cyclopentyl-5-(4-methoxy-phenyl)-7H-pyrrolo[2,3-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of p60 c-Src tyrosine kinase mediated phosphorylation of Fak in IC8.1 fibroblastsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3RMFPubMed
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