Compile Data Set for Download or QSAR

Found 59 hits of Enzyme Inhibition Constant Data   

TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)copy SMILEScopy InChI
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)copy SMILEScopy InChI
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  0.520nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)copy SMILEScopy InChI
Affinity DataKi:  0.720nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.760nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  0.780nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.830nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  1.23nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  1.51nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  2.14nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  2.63nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)copy SMILEScopy InChI
Affinity DataKi:  4.07nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  4.68nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  4.90nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  9.55nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)copy SMILEScopy InChI
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  13.2nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  13.8nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  17.4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  41.7nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  42.7nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  49.0nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  53.7nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  56.2nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  83.2nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)copy SMILEScopy InChI
Affinity DataKi:  110nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)copy SMILEScopy InChI
Affinity DataKi:  132nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  214nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  219nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  224nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)copy SMILEScopy InChI
Affinity DataKi:  229nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Pharma AG

Curated by PDSP Ki Database
LigandPNGBDBM82467(2-Deamino-L-Abu(1)-L-Lys-L-Asp(NH2)-L-Phe-L-Phe-L-...)copy SMILEScopy InChI
Affinity DataKi:  257nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7DTQPubMed
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