Found 17 hits of Enzyme Inhibition Constant Data
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.5nMAssay Description:Binding affinity to VEGFR2More data for this Ligand-Target Pair
Affinity DataKd: 5.30nMAssay Description:Binding affinity to PKN1More data for this Ligand-Target Pair
TargetPhosphorylase b kinase gamma catalytic chain, liver/testis isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 5.90nMAssay Description:Binding affinity to PHKG2More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity to YSK1More data for this Ligand-Target Pair
Affinity DataKd: 540nMAssay Description:Binding affinity to BRAFMore data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding affinity to MST3More data for this Ligand-Target Pair
Affinity DataKd: 340nMAssay Description:Binding affinity to MST4More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding affinity to HPK1More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 59nMAssay Description:Binding affinity to VEGFR2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CDK2More data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Binding affinity to CDK11More data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding affinity to CDK8More data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Binding affinity to p38-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 2.40E+3nMAssay Description:Binding affinity to PAK6More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Binding affinity to DYRK1AMore data for this Ligand-Target Pair
Affinity DataKd: 3.70nMAssay Description:Binding affinity to JH1 catalytic domain JAK2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TGFBR1More data for this Ligand-Target Pair
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