Found 1 hit of Enzyme Inhibition Constant Data
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University of Shizuoka
Curated by ChEMBL
University of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Antagonist activity against human TRPV1 expressed in T-REx HEK cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ accum...More data for this Ligand-Target Pair