Found 1 hit of Enzyme Inhibition Constant Data
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University in Saint Louis
Curated by ChEMBL
Washington University in Saint Louis
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair