Compile Data Set for Download or QSAR

Found 3 hits of Enzyme Inhibition Constant Data   

LigandPNGBDBM50438224(CHEMBL2407759)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
OSI Pharmaceuticals LLC

Curated by ChEMBL
LigandPNGBDBM50438224(CHEMBL2407759)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of TAK1 in human HCT116 cells assessed as inhibition of TNF-alpha-stimulated JNK phosphorylationMore data for this Ligand-Target Pair
LigandPNGBDBM50438225(CHEMBL2407766)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATPMore data for this Ligand-Target Pair
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