Compile Data Set for Download or QSAR

Found 31 hits of Enzyme Inhibition Constant Data   

TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215536((R)-Alpha-Methylhistamine | CHEBI:73337 | CHEMBL26...)copy SMILEScopy InChI
Affinity DataKi:  0.0851nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)copy SMILEScopy InChI
Affinity DataKi:  0.145nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215536((R)-Alpha-Methylhistamine | CHEBI:73337 | CHEMBL26...)copy SMILEScopy InChI
Affinity DataKi:  0.151nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215541(CHEMBL299589)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215541(CHEMBL299589)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215548(CHEMBL301176)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50216735(CHEMBL55836)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215549(CHEMBL53361)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50216734(CHEMBL300704)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215548(CHEMBL301176)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215543(CHEMBL55018)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215539(CHEMBL417017)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50216734(CHEMBL300704)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215539(CHEMBL417017)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215549(CHEMBL53361)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215543(CHEMBL55018)copy SMILEScopy InChI
Affinity DataKi:  38nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215538(CHEMBL52090)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215538(CHEMBL52090)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50216733(CHEMBL52080)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215537(CHEMBL54858)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50216736(CHEMBL53412)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215544(CHEMBL298581)copy SMILEScopy InChI
Affinity DataKi:  107nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50216733(CHEMBL52080)copy SMILEScopy InChI
Affinity DataKi:  115nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50216736(CHEMBL53412)copy SMILEScopy InChI
Affinity DataKi:  138nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215537(CHEMBL54858)copy SMILEScopy InChI
Affinity DataKi:  186nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215542(CHEMBL301838)copy SMILEScopy InChI
Affinity DataKi:  490nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215544(CHEMBL298581)copy SMILEScopy InChI
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215542(CHEMBL301838)copy SMILEScopy InChI
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215540(CHEMBL53056)copy SMILEScopy InChI
Affinity DataKi:  1.86E+3nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
TargetHistamine H3 receptor(GUINEA PIG)
The James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50215540(CHEMBL53056)copy SMILEScopy InChI
Affinity DataKi:  2.88E+3nMAssay Description:Binding affinity towards histamine H3 receptor using [3H](R)-alpha-methylhistamine as radioligand in guinea pig ileum LMMP homogenatesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24T6MKGPubMed
* indicates data uncertainty>20%