Compile Data Set for Download or QSAR

Found 63 hits of Enzyme Inhibition Constant Data   

TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50051753(1-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-yl)...)copy SMILEScopy InChI
Affinity DataKi:  0.230nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099228(1-[3-(6-Iodo-naphthalen-2-yl)-8-methyl-8-aza-bicyc...)copy SMILEScopy InChI
Affinity DataKi:  0.370nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099227(1-[3-(6-Ethyl-naphthalen-2-yl)-8-methyl-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataKi:  0.380nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099223(1-[3-(7-Iodo-naphthalen-2-yl)-8-methyl-8-aza-bicyc...)copy SMILEScopy InChI
Affinity DataKi:  0.470nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041304(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  1.06nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099233(1-[3-(6-Isopropyl-naphthalen-2-yl)-8-methyl-8-aza-...)copy SMILEScopy InChI
Affinity DataKi:  1.97nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50051753(1-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-yl)...)copy SMILEScopy InChI
Affinity DataKi:  2.05nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099225(2-Methyl-1-(8-methyl-3-naphthalen-2-yl-8-aza-bicyc...)copy SMILEScopy InChI
Affinity DataKi:  2.08nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099235(1-[3-(6-Methoxy-naphthalen-2-yl)-8-methyl-8-aza-bi...)copy SMILEScopy InChI
Affinity DataKi:  2.24nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099222(1-[3-(5-Iodo-6-methoxy-naphthalen-2-yl)-8-methyl-8...)copy SMILEScopy InChI
Affinity DataKi:  2.27nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041304(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099231(1-[3-(5-Ethyl-6-methoxy-naphthalen-2-yl)-8-methyl-...)copy SMILEScopy InChI
Affinity DataKi:  7.55nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099226(1-[8-Methyl-3-(4-methyl-naphthalen-1-yl)-8-aza-bic...)copy SMILEScopy InChI
Affinity DataKi:  8.99nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099230(1-[3-(6-Methoxy-5-nitro-naphthalen-2-yl)-8-methyl-...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099229(1-[3-(5-Acetyl-6-methoxy-naphthalen-2-yl)-8-methyl...)copy SMILEScopy InChI
Affinity DataKi:  15.8nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  16.4nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  16.4nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041300(1-(8-Methyl-3-naphthalen-1-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041298(1-(8-Methyl-3-naphthalen-1-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041298(1-(8-Methyl-3-naphthalen-1-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099227(1-[3-(6-Ethyl-naphthalen-2-yl)-8-methyl-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataKi:  27.7nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041303(1-[3-(4-Isopropyl-phenyl)-8-methyl-8-aza-bicyclo[3...)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099225(2-Methyl-1-(8-methyl-3-naphthalen-2-yl-8-aza-bicyc...)copy SMILEScopy InChI
Affinity DataKi:  37.6nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041300(1-(8-Methyl-3-naphthalen-1-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041296(1-(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct-2-yl...)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099234(1-[3-(5-Isopropenyl-6-methoxy-naphthalen-2-yl)-8-m...)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041296(1-(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct-2-yl...)copy SMILEScopy InChI
Affinity DataKi:  131nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099232(1-[3-(4-Isopropyl-naphthalen-1-yl)-8-methyl-8-aza-...)copy SMILEScopy InChI
Affinity DataKi:  136nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099226(1-[8-Methyl-3-(4-methyl-naphthalen-1-yl)-8-aza-bic...)copy SMILEScopy InChI
Affinity DataKi:  163nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041298(1-(8-Methyl-3-naphthalen-1-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataKi:  165nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099224(1-[3-(4-Ethyl-naphthalen-1-yl)-8-methyl-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataKi:  175nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to serotonin transporter (SERT) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099229(1-[3-(5-Acetyl-6-methoxy-naphthalen-2-yl)-8-methyl...)copy SMILEScopy InChI
Affinity DataKi:  498nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099222(1-[3-(5-Iodo-6-methoxy-naphthalen-2-yl)-8-methyl-8...)copy SMILEScopy InChI
Affinity DataKi:  781nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099234(1-[3-(5-Isopropenyl-6-methoxy-naphthalen-2-yl)-8-m...)copy SMILEScopy InChI
Affinity DataKi:  2.33E+3nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099231(1-[3-(5-Ethyl-6-methoxy-naphthalen-2-yl)-8-methyl-...)copy SMILEScopy InChI
Affinity DataKi:  3.36E+3nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099224(1-[3-(4-Ethyl-naphthalen-1-yl)-8-methyl-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataKi:  4.77E+3nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099232(1-[3-(4-Isopropyl-naphthalen-1-yl)-8-methyl-8-aza-...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetTransporter(Rattus norvegicus)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041303(1-[3-(4-Isopropyl-phenyl)-8-methyl-8-aza-bicyclo[3...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Affinity for the displacement of [3H]-paroxetine binding to norepinephrine transporter (NET) in rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50051753(1-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 0.0300nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099235(1-[3-(6-Methoxy-naphthalen-2-yl)-8-methyl-8-aza-bi...)copy SMILEScopy InChI
Affinity DataIC50: 0.130nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099227(1-[3-(6-Ethyl-naphthalen-2-yl)-8-methyl-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099225(2-Methyl-1-(8-methyl-3-naphthalen-2-yl-8-aza-bicyc...)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099228(1-[3-(6-Iodo-naphthalen-2-yl)-8-methyl-8-aza-bicyc...)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099233(1-[3-(6-Isopropyl-naphthalen-2-yl)-8-methyl-8-aza-...)copy SMILEScopy InChI
Affinity DataIC50: 0.390nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099223(1-[3-(7-Iodo-naphthalen-2-yl)-8-methyl-8-aza-bicyc...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041304(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataIC50: 1.27nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50099222(1-[3-(5-Iodo-6-methoxy-naphthalen-2-yl)-8-methyl-8...)copy SMILEScopy InChI
Affinity DataIC50: 1.31nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataIC50: 2.51nMAssay Description:Inhibitory activity in displacing [125I]- RTI-55 binding to dopamine transporter in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H1318RPubMed
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