Found 71 hits of Enzyme Inhibition Constant Data
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program/NIH
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Ability to displace [3H]-WIN-35,428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair