Compile Data Set for Download or QSAR

Found 5 hits of Enzyme Inhibition Constant Data   

TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)copy SMILEScopy InChI
Affinity DataKi:  0.251nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50473964(CHEMBL2370836)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50473965(CHEMBL2370837)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
* indicates data uncertainty>20%