Compile Data Set for Download or QSAR

Found 61 hits of Enzyme Inhibition Constant Data   

TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137141(4-Chloro-2-[3-(1H-indol-2-yl)-ureido]-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137159(4-Chloro-2-[3-(3-chloro-phenyl)-ureido]-benzoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137133(4,6-Bis-benzoylamino-isophthalic acid | CHEMBL1567...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137142(2-[3-(4-Bromo-phenyl)-ureido]-4-chloro-benzoic aci...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137129(4-Chloro-2-[3-(3-iodo-phenyl)-ureido]-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137157(4-Chloro-2-[3-(4-chloro-phenyl)-ureido]-benzoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137169(2-(3-Benzo[1,3]dioxol-5-yl-ureido)-4-chloro-benzoi...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137145(4-Chloro-2-[3-(3-methoxy-phenyl)-ureido]-benzoic a...)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137153(2-[3-(2-Bromo-phenyl)-ureido]-4-chloro-benzoic aci...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137150(4-Chloro-2-[3-(2-trifluoromethyl-phenyl)-ureido]-b...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137128(4-Chloro-2-[3-(2-chloro-phenyl)-ureido]-benzoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137164(4-Chloro-2-[3-(4-iodo-phenyl)-ureido]-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137125(2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137136(4-Chloro-2-[3-(4-trifluoromethyl-phenyl)-ureido]-b...)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137131(4-Chloro-2-[3-(2-iodo-phenyl)-ureido]-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137149(4-Chloro-2-[3-(3-trifluoromethyl-phenyl)-ureido]-b...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137143(4-Bromo-2-[3-(3-trifluoromethyl-phenyl)-ureido]-be...)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137138(4-Chloro-2-[3-(3-fluoro-phenyl)-ureido]-benzoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137147(4-Chloro-2-(3-naphthalen-1-yl-ureido)-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 9.40E+3nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137166(4-Fluoro-2-[3-(3-trifluoromethyl-phenyl)-ureido]-b...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137170(2-(3-Biphenyl-2-yl-ureido)-4-chloro-benzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137140(4-Chloro-2-(3-phenyl-ureido)-benzoic acid | CHEMBL...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137130(4-Chloro-2-[3-(4-methoxy-phenyl)-ureido]-benzoic a...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137144(2-(3-Biphenyl-3-yl-ureido)-4-chloro-benzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137158(4-Chloro-2-[3-(2-methoxy-phenyl)-ureido]-benzoic a...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137134(4-Chloro-2-[3-(4-fluoro-phenyl)-ureido]-benzoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137168(4-Chloro-2-[3-(3-hydroxy-phenyl)-ureido]-benzoic a...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137165(4-Chloro-2-(3-thiophen-2-yl-ureido)-benzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137162(4-Chloro-2-[3-(2-fluoro-phenyl)-ureido]-benzoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137160(4-Chloro-2-[3-(2-hydroxy-phenyl)-ureido]-benzoic a...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137151(4-Trifluoromethyl-2-[3-(3-trifluoromethyl-phenyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137125(2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+4nMAssay Description:In vitro inhibitory activity of the compound against Ionotropic glutamate receptor ionotropic kainate 2 (GluR-6) of HEK293 cells in FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137137(2-(3-Biphenyl-4-yl-ureido)-4-chloro-benzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137127(4-Nitro-2-[3-(3-trifluoromethyl-phenyl)-ureido]-be...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137125(2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Binding inhibition of compound against Ionotropic glutamate receptor ionotropic kainate 1 (GluR5) using [3H]-ATPA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137124(4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Binding inhibition of compound against Ionotropic glutamate receptor ionotropic kainate 1 (GluR5) using [3H]-ATPA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137167(2-(3-Anthracen-2-yl-ureido)-4-chloro-benzoic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137126(4-Methyl-2-[3-(3-trifluoromethyl-phenyl)-ureido]-b...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137152(4-Chloro-2-(3-pyridin-2-yl-ureido)-benzoic acid | ...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137156(4-Chloro-2-[3-(4-hydroxy-phenyl)-ureido]-benzoic a...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137135(4-Chloro-2-(3-thiophen-3-yl-ureido)-benzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137132(3-[3-(3-Trifluoromethyl-phenyl)-ureido]-naphthalen...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137124(4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+4nMAssay Description:In vitro inhibitory activity of the compound against Ionotropic glutamate receptor ionotropic kainate 2 (GluR-6) of HEK293 cells in FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137124(4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137124(4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137146(4-Chloro-2-(3-pyridin-3-yl-ureido)-benzoic acid | ...)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137154(2-[3-(3-Trifluoromethyl-phenyl)-ureido]-benzoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 7.20E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137161(4-Chloro-2-(3-pyridin-4-yl-ureido)-benzoic acid | ...)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+4nMAssay Description:In vitro inhibitory activity against human ionotropic glutamate receptor ionotropic kainate 1 (GluR-5) expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137125(2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity of the compound against Ionotropic glutamate receptor AMPA 4 of HEK293 cells in FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50137124(4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity of the compound against Ionotropic glutamate receptor AMPA 1 of HEK293 cells in FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9B60PubMed
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