Compile Data Set for Download or QSAR

Found 5 hits of Enzyme Inhibition Constant Data   

TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50072394(1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyr...)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]-[3-Me-His2]-TRH binding to thyrotropin releasing hormone receptor of rat forebrainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095F0PubMed
TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50156181(3-carbamoyl-1-{3-(2-carbamoyl-pyrrolidin-1-yl)-3-o...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-[3-Me-His2]-TRH binding to thyrotropin releasing hormone receptor of rat forebrainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095F0PubMed
TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50156183(3-carbamoyl-1-{6-(2-carbamoyl-pyrrolidin-1-yl)-6-o...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-[3-Me-His2]-TRH binding to thyrotropin releasing hormone receptor of rat forebrainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095F0PubMed
TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50156179(3-carbamoyl-1-{4-(2-carbamoyl-pyrrolidin-1-yl)-4-o...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-[3-Me-His2]-TRH binding to thyrotropin releasing hormone receptor of rat forebrainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095F0PubMed
TargetThyrotropin-releasing hormone receptor(Rattus norvegicus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50156182(3-carbamoyl-1-{5-(2-carbamoyl-pyrrolidin-1-yl)-5-o...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-[3-Me-His2]-TRH binding to thyrotropin releasing hormone receptor of rat forebrainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095F0PubMed
* indicates data uncertainty>20%