Compile Data Set for Download or QSAR

Found 3 hits of Enzyme Inhibition Constant Data   

TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50137962((1R,2S)-1-((3R,5S)-1-((S)-2-((S)-2-acetamido-2-cyc...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human leucocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C1WCSPubMed
TargetCathepsin B(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50137962((1R,2S)-1-((3R,5S)-1-((S)-2-((S)-2-acetamido-2-cyc...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C1WCSPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50157704((1R,2S)-1-((3R,5S)-1-((S)-2-(tert-butoxycarbonyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of human leucocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C1WCSPubMed
* indicates data uncertainty>20%