Compile Data Set for Download or QSAR

Found 9 hits of Enzyme Inhibition Constant Data   

TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161249(3a,11a-dihydroxy-4''-imino-9,15a-dimethyl-1-(5-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161262(11a-hydroxy-3a,13a-di(hydroxymethyl)-9,15a-dimethy...)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161244(CHEMBL369515 | Uscharin derivative)copy SMILEScopy InChI
Affinity DataIC50: 1.89E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161268(CHEMBL366906 | Uscharin derivative)copy SMILEScopy InChI
Affinity DataIC50: 4.08E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161245(11a-hydroxy-3a-hydroxymethyl-4''-imino-9,15a-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 1.21E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161252(CHEMBL427124 | Uscharin derivative)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161246(11a-hydroxy-3a-hydroxymethyl-4''-imino-9,15a-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161272(CHEMBL262795 | Uscharin derivative)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen SA

Curated by ChEMBL
LigandPNGBDBM50161253(CHEMBL426228 | Uscharin derivative)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0SD1PubMed
* indicates data uncertainty>20%