Compile Data Set for Download or QSAR

Found 56 hits of Enzyme Inhibition Constant Data   

TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84541(Indirubin derivative, 22)copy SMILEScopy InChI
Affinity DataIC50: 10nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84539(Indirubin derivative, 36 (X=O))copy SMILEScopy InChI
Affinity DataIC50: 20nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84542(Indirubin derivative, 23)copy SMILEScopy InChI
Affinity DataIC50: 40nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84555(Indirubin derivative, 30a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 40nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84535(Indirubin derivative, 8)copy SMILEScopy InChI
Affinity DataIC50: 40nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84536(Indirubin derivative, 32)copy SMILEScopy InChI
Affinity DataIC50: 40nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84546(Indirubin derivative, 27a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 70nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 70nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84537(Indirubin derivative, 33)copy SMILEScopy InChI
Affinity DataIC50: 80nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)copy SMILEScopy InChI
Affinity DataIC50: 80nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84544(Indirubin derivative, 36 (X=NO))copy SMILEScopy InChI
Affinity DataIC50: 80nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84548(Indirubin derivative, 29a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 90nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84543(Indirubin derivative, 25)copy SMILEScopy InChI
Affinity DataIC50: 90nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84534(Indirubin derivative, 20)copy SMILEScopy InChI
Affinity DataIC50: 300nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 400nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84540(Indirubin derivative, 35)copy SMILEScopy InChI
Affinity DataIC50: 450nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84534(Indirubin derivative, 20)copy SMILEScopy InChI
Affinity DataIC50: 500nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84555(Indirubin derivative, 30a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 600nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84546(Indirubin derivative, 27a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 600nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84538(Indirubin derivative, 34)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84552(Indirubin derivative, 37)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM7392(2-[(3Z)-2-oxo-2,3-dihydro-1H-indol-3-ylidene]-2,3-...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84545(Indirubin derivative, 26)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84550(Indirubin derivative, 31a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84536(Indirubin derivative, 32)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84548(Indirubin derivative, 29a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetInsulin receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84555(Indirubin derivative, 30a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetInsulin receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84534(Indirubin derivative, 20)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetKit ligand(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84555(Indirubin derivative, 30a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetInsulin receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84550(Indirubin derivative, 31a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetKit ligand(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84534(Indirubin derivative, 20)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84555(Indirubin derivative, 30a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetKit ligand(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetInsulin receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetInsulin receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84534(Indirubin derivative, 20)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetKit ligand(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84555(Indirubin derivative, 30a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84555(Indirubin derivative, 30a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetKit ligand(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84553(Indirubin derivative, 28a | Indirubin derivative, ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetKit ligand(Homo sapiens (Human))
Schering AG

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM84534(Indirubin derivative, 20)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Schering AG

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMpH: 7.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56H8HPubMed
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