Found 58 hits of Enzyme Inhibition Constant Data
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataKi: 8.80E+3nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataKi: 9.00E+3nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Antiproliferative activity against human NPM-ALK positive anaplastic large cell lymphoma karpas299 cell lineMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Antiproliferative activity against human BCR-ABL positive chronic myeloid leukemia K562 cell lineMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against Flt3More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity against Flt3More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Antiproliferative activity against murine BaF3 cell line expressing NPM-ALKMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against IGF1RMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Antiproliferative activity against human NPM-ALK positive anaplastic large cell lymphoma karpas299 cell lineMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 9.40E+3nMAssay Description:Antiproliferative activity against human NPM-ALK positive anaplastic large cell lymphoma karpas299 cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Antiproliferative activity against human BCR-ABL positive chronic myeloid leukemia K562 cell lineMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Antiproliferative activity against human NPM-ALK positive anaplastic large cell lymphoma karpas299 cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.29E+4nMAssay Description:Antiproliferative activity against human BCR-ABL positive chronic myeloid leukemia K562 cell lineMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Antiproliferative activity against murine BaF3 cell line expressing NPM-ALKMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.46E+4nMAssay Description:Antiproliferative activity against human BCR-ABL positive chronic myeloid leukemia K562 cell lineMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against IGF1RMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.74E+4nMAssay Description:Antiproliferative activity against murine BaF3 cell line expressing NPM-ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against IGF1RMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against AblMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against SrcMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against AblMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Flt3More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against SrcMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against AblMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against SrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against SrcMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against AblMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against IGF1RMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Flt3More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.03E+4nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Antiproliferative activity against murine BaF3 cell line expressing NPM-ALKMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 2.73E+4nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair