Compile Data Set for Download or QSAR

Found 5 hits of Enzyme Inhibition Constant Data   

TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50248765(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of His6-tagged RSK2 C-terminal domian expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8Z60PubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50324685(2-(3-(4-amino-6-(2-fluoroacetyl)-5-p-tolyl-7H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of His6-tagged RSK2 C-terminal domian expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8Z60PubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50324684(3-(1-(4-amino-6-(2-fluoroacetyl)-5-p-tolyl-7H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His6-tagged RSK2 C-terminal domian expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8Z60PubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50248765(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)copy SMILEScopy InChI
Affinity DataEC50:  150nMAssay Description:Inhibition of PMA-stimulated RSK2 phosphorylation in HEK293 cells after 1 hr by western blotting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8Z60PubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50324684(3-(1-(4-amino-6-(2-fluoroacetyl)-5-p-tolyl-7H-pyrr...)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of PMA-stimulated RSK2 phosphorylation in HEK293 cells after 1 hr by western blotting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B8Z60PubMed
* indicates data uncertainty>20%