Found 84 hits of Enzyme Inhibition Constant Data
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 9.40nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 11.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 15.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 16.2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 21.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 29.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 33.4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 51.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 82.7nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 88.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 94.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 142nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 162nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 197nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 198nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 298nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 495nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 552nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 708nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 775nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataEC50: 39.5nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataEC50: 33.8nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataEC50: 285nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataEC50: 392nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University of Minnesota Health Science Center
Curated by ChEMBL
University of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataEC50: 91.7nMAssay Description:Activity at metastin receptor expressed in HEK293 cells by measuring calcium releaseMore data for this Ligand-Target Pair