Found 29 hits of Enzyme Inhibition Constant Data
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 175nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 408nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 432nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 2.99E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 6.69E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
TargetProtein kinase C beta type(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PKCbetaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SykMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ZAPMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Kissei Pharmaceutical Company Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair