Compile Data Set for Download or QSAR

Found 29 hits of Enzyme Inhibition Constant Data   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375360(CHEMBL261188)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375361(CHEMBL260157)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375366(CHEMBL406418)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375364(CHEMBL261743)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375362(CHEMBL260860)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375363(CHEMBL261744)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375367(CHEMBL405893)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375368(CHEMBL259200)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375365(CHEMBL261450)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375360(CHEMBL261188)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375366(CHEMBL406418)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375356(CHEMBL260114)copy SMILEScopy InChI
Affinity DataIC50: 175nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375358(CHEMBL258677)copy SMILEScopy InChI
Affinity DataIC50: 408nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375369(CHEMBL260024)copy SMILEScopy InChI
Affinity DataIC50: 432nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375361(CHEMBL260157)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375356(CHEMBL260114)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of human cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375370(CHEMBL410296)copy SMILEScopy InChI
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375357(CHEMBL412139)copy SMILEScopy InChI
Affinity DataIC50: 2.99E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375371(CHEMBL412273)copy SMILEScopy InChI
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375359(CHEMBL427741)copy SMILEScopy InChI
Affinity DataIC50: 6.69E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375372(CHEMBL259627)copy SMILEScopy InChI
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of human cSrcMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PKCbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SykMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ZAPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kissei Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50375355(CHEMBL260861)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9R01PubMed
* indicates data uncertainty>20%