Found 62 hits of Enzyme Inhibition Constant Data
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 93nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 123nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 141nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 302nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 302nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 309nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 331nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 331nMAssay Description:Displacement of [3]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 372nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 372nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 398nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 398nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 398nMAssay Description:Displacement of [3]ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 427nMAssay Description:Displacement of [3]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Santiago de Compostela
Curated by ChEMBL
University of Santiago de Compostela
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of [3]NECA from human adenosine A3 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair