Compile Data Set for Download or QSAR

Found 124 hits of Enzyme Inhibition Constant Data   

TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376975(CHEMBL260570)copy SMILEScopy InChI
Affinity DataKi:  0.450nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM23617((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-nitrophe...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376976(CHEMBL261227)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376971(CHEMBL438046)copy SMILEScopy InChI
Affinity DataKi:  18.9nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376977(CHEMBL408670)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376974(CHEMBL261226)copy SMILEScopy InChI
Affinity DataKi:  300nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376972(CHEMBL259855)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376970(CHEMBL258729)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376973(CHEMBL260281)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412033(CHEMBL260688)copy SMILEScopy InChI
Affinity DataIC50: 2.75nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412008(CHEMBL259866)copy SMILEScopy InChI
Affinity DataIC50: 4.79nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376975(CHEMBL260570)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM23617((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-nitrophe...)copy SMILEScopy InChI
Affinity DataIC50: 8.51nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411998(CHEMBL265689)copy SMILEScopy InChI
Affinity DataIC50: 15.8nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50222744((2R,3R,4S,5R)-2-(6-(4-nitrobenzylthio)-2-amino-9H-...)copy SMILEScopy InChI
Affinity DataIC50: 21.4nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411987(CHEMBL260055)copy SMILEScopy InChI
Affinity DataIC50: 21.9nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411986(CHEMBL260166)copy SMILEScopy InChI
Affinity DataIC50: 27.5nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412000(CHEMBL410278)copy SMILEScopy InChI
Affinity DataIC50: 31.6nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412042(CHEMBL260882)copy SMILEScopy InChI
Affinity DataIC50: 33.1nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412004(CHEMBL260645)copy SMILEScopy InChI
Affinity DataIC50: 69.2nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412017(CHEMBL409320)copy SMILEScopy InChI
Affinity DataIC50: 77.6nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412007(CHEMBL408710)copy SMILEScopy InChI
Affinity DataIC50: 81.3nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411995(CHEMBL258627)copy SMILEScopy InChI
Affinity DataIC50: 87.1nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411988(CHEMBL411899)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412003(CHEMBL410465)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412048(CHEMBL265930)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412049(CHEMBL411065)copy SMILEScopy InChI
Affinity DataIC50: 178nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412056(CHEMBL263651)copy SMILEScopy InChI
Affinity DataIC50: 178nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376976(CHEMBL261227)copy SMILEScopy InChI
Affinity DataIC50: 182nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411990(CHEMBL261793)copy SMILEScopy InChI
Affinity DataIC50: 182nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412010(CHEMBL259303)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412013(CHEMBL259759)copy SMILEScopy InChI
Affinity DataIC50: 224nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412009(CHEMBL259301)copy SMILEScopy InChI
Affinity DataIC50: 245nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412005(CHEMBL411710)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412050(CHEMBL259189)copy SMILEScopy InChI
Affinity DataIC50: 282nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412051(CHEMBL261528)copy SMILEScopy InChI
Affinity DataIC50: 282nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411979(CHEMBL427558)copy SMILEScopy InChI
Affinity DataIC50: 309nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412011(CHEMBL412113)copy SMILEScopy InChI
Affinity DataIC50: 331nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50376971(CHEMBL438046)copy SMILEScopy InChI
Affinity DataIC50: 331nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411999(CHEMBL261664)copy SMILEScopy InChI
Affinity DataIC50: 347nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412014(CHEMBL261530)copy SMILEScopy InChI
Affinity DataIC50: 355nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412012(CHEMBL411687)copy SMILEScopy InChI
Affinity DataIC50: 363nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412073(CHEMBL412078)copy SMILEScopy InChI
Affinity DataIC50: 427nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412062(CHEMBL294755)copy SMILEScopy InChI
Affinity DataIC50: 457nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412002(CHEMBL261887)copy SMILEScopy InChI
Affinity DataIC50: 617nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411992(CHEMBL261327)copy SMILEScopy InChI
Affinity DataIC50: 708nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412069(CHEMBL409354)copy SMILEScopy InChI
Affinity DataIC50: 813nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412006(CHEMBL408449)copy SMILEScopy InChI
Affinity DataIC50: 813nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50411994(CHEMBL410084)copy SMILEScopy InChI
Affinity DataIC50: 977nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50412059(CHEMBL260497)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8866PubMed
Displayed 1 to 50 (of 124 total ) | Next | Last >>* indicates data uncertainty>20%