Found 124 hits of Enzyme Inhibition Constant Data
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 18.9nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of 5-(SAENTA)-X8-fluorescein from human ENT1 transporter in human K562 cellsMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 2.75nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 4.79nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 8.51nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 15.8nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 21.4nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 21.9nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 27.5nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 31.6nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 33.1nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 69.2nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 77.6nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 81.3nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 87.1nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 123nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 178nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 178nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 182nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 182nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 245nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 282nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 282nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 309nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 331nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 331nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 347nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 355nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 363nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 427nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 457nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 617nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 708nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 813nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 813nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 977nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center
Curated by ChEMBL
University of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair