Compile Data Set for Download or QSAR

Found 8 hits of Enzyme Inhibition Constant Data   

TargetTGF-beta receptor type-1(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50272008(1-{2-[(6,7-dimethoxy-4-quinolyl)oxy]-4,5-dimethylp...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of ALK5 (unknown origin) by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50271724(CHEMBL482729 | {2-[(6,7-Dimethoxy-4-quinolyl)oxy]-...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50271724(CHEMBL482729 | {2-[(6,7-Dimethoxy-4-quinolyl)oxy]-...)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of ALK5 (unknown origin) by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50271837(1-{2-[(6,7-dimethoxy-4-quinolyl)oxy]-5-methylpheny...)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of ALK5 (unknown origin) by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50271723(CHEMBL482728 | {2-[(6,7-Dimethoxy-4-quinolyl)oxy]p...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50271837(1-{2-[(6,7-dimethoxy-4-quinolyl)oxy]-5-methylpheny...)copy SMILEScopy InChI
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50272008(1-{2-[(6,7-dimethoxy-4-quinolyl)oxy]-4,5-dimethylp...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
KIRIN Pharma Co Ltd

Curated by ChEMBL
LigandPNGBDBM50271723(CHEMBL482728 | {2-[(6,7-Dimethoxy-4-quinolyl)oxy]p...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of ALK5 (unknown origin) by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22807D8PubMed
* indicates data uncertainty>20%