Found 72 hits of Enzyme Inhibition Constant Data
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 1.72nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 1.77nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 2.38nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 3.26nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 3.45nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 4.28nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 5.36nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 5.57nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 6.71nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 6.92nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 9.36nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 14.9nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 15.1nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 21.7nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 28.1nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 33.4nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 33.5nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 36.6nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 45.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 50.8nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 51.3nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 56.6nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 81.8nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 83.4nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 87.3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 87.4nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 88.3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 97.7nMAssay Description:Displacement of [3H]WIN-35428 from DAT in rat striatum membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 235nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 246nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 273nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 292nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 318nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 497nMAssay Description:Displacement of [3H]nisoxetine from NET in rat frontal cortex membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 521nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 543nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 766nMAssay Description:Displacement of [3H]nisoxetine from NET in rat frontal cortex membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 779nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 803nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetTransporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 810nMAssay Description:Displacement of [3H]nisoxetine from NET in rat frontal cortex membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 835nMAssay Description:Displacement of [3H]citalopram from SERT in rat brain stem membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute on Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 893nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair