Compile Data Set for Download or QSAR

Found 30 hits of Enzyme Inhibition Constant Data   

TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  570nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  1.16E+3nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)copy SMILEScopy InChI
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254389((2S)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi:  5.90E+4nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254338((2R)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi:  2.10E+5nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254389((2S)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi:  2.93E+5nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254391((2S)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254391((2S)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254337((2S)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254390((2R)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254338((2R)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi:  3.36E+5nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254392((2R)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254337((2S)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254390((2R)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254390((2R)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254391((2S)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254338((2R)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254392((2R)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254392((2R)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254389((2S)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254337((2S)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50007548((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254390((2R)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254389((2S)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254337((2S)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Salerno

Curated by ChEMBL
LigandPNGBDBM50254338((2R)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine | C...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7WKFPubMed
* indicates data uncertainty>20%