Found 24 hits of Enzyme Inhibition Constant Data
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of CSF1R (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of PDGFRb (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 478nMAssay Description:Inhibition of PTK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 672nMAssay Description:Inhibition of EphB4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of IGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Jnk1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Plk (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Kdr (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Cdk2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Pak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Csk (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
AstraZeneca R&D Boston
Curated by ChEMBL
AstraZeneca R&D Boston
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Chk1 (unknown origin)More data for this Ligand-Target Pair