Compile Data Set for Download or QSAR

Found 198 hits of Enzyme Inhibition Constant Data   

TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  0.580nMAssay Description:Binding affinity to thromboxane receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333841((R)-2-(3,4-difluoro-7-(4-fluoro-N-methylphenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333868((R)-2-(3-fluoro-7-(4-fluoro-N-methylphenylsulfonam...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333869((R)-2-(3-chloro-7-(4-fluoro-N-methylphenylsulfonam...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333850((R)-2-(7-(4-fluoro-N-(4-fluorobenzyl)phenylsulfona...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50161745(CHEMBL179036 | {3-[((R)-4-Fluoro-benzenesulfonyl)-...)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333844((R)-2-(4-fluoro-7-(4-fluoro-N-methylphenylsulfonam...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333848((R)-2-(7-(4-fluoro-N-pentylphenylsulfonamido)-6,7,...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333870((R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-3-(t...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333847((R)-2-(7-(N-ethyl-4-fluorophenylsulfonamido)-6,7,8...)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333872((R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-3-ph...)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50296980((R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-6,7,...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333876((R)-2-(2,3-difluoro-7-(4-fluoro-N-methylphenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333843((R)-2-(3-chloro-2-fluoro-7-(4-fluoro-N-methylpheny...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333851((R)-2-(7-(4-fluoro-N-(2,2,2-trifluoroethyl)phenyls...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333845((R)-2-(2,4-difluoro-7-(4-fluoro-N-methylphenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333856((R)-2-(7-(N-methylphenylsulfonamido)-6,7,8,9-tetra...)copy SMILEScopy InChI
Affinity DataKi:  4.30nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333864((R)-2-(7-(4-methoxy-N-methylphenylsulfonamido)-6,7...)copy SMILEScopy InChI
Affinity DataKi:  4.40nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333867((R)-2-(2-fluoro-7-(4-fluoro-N-methylphenylsulfonam...)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333849((R)-2-(7-(N-(cyclopropylmethyl)-4-fluorophenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333857((R)-2-(7-(4-chloro-N-methylphenylsulfonamido)-6,7,...)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333842((R)-2-(1,3-dichloro-7-(4-fluoro-N-methylphenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  5.60nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50161745(CHEMBL179036 | {3-[((R)-4-Fluoro-benzenesulfonyl)-...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333861((R)-2-(7-(5-chloro-N-methylthiophene-2-sulfonamido...)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333853((R)-2-(7-(N,2-dimethylphenylsulfonamido)-6,7,8,9-t...)copy SMILEScopy InChI
Affinity DataKi:  7.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333855((R)-2-(7-(N,3-dimethylphenylsulfonamido)-6,7,8,9-t...)copy SMILEScopy InChI
Affinity DataKi:  8.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333875((R)-2-(3-cyano-7-(4-fluoro-N-methylphenylsulfonami...)copy SMILEScopy InChI
Affinity DataKi:  8.80nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333846((R)-2-(7-(4-fluorophenylsulfonamido)-6,7,8,9-tetra...)copy SMILEScopy InChI
Affinity DataKi:  9.80nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333873((R)-2-(1-fluoro-7-(4-fluoro-N-methylphenylsulfonam...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333846((R)-2-(7-(4-fluorophenylsulfonamido)-6,7,8,9-tetra...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Binding affinity to thromboxane receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333871((R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-3-(m...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333847((R)-2-(7-(N-ethyl-4-fluorophenylsulfonamido)-6,7,8...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333851((R)-2-(7-(4-fluoro-N-(2,2,2-trifluoroethyl)phenyls...)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333859((R)-2-(7-(4-ethyl-N-methylphenylsulfonamido)-6,7,8...)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333852((R)-2-(7-(2-fluoro-N-methylphenylsulfonamido)-6,7,...)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333860((R)-2-(7-(1-(4-fluorophenyl)-N-methylmethylsulfona...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333859((R)-2-(7-(4-ethyl-N-methylphenylsulfonamido)-6,7,8...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333854((R)-2-(7-(3-fluoro-N-methylphenylsulfonamido)-6,7,...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333842((R)-2-(1,3-dichloro-7-(4-fluoro-N-methylphenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333864((R)-2-(7-(4-methoxy-N-methylphenylsulfonamido)-6,7...)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333858((R)-2-(7-(N-methyl-4-(trifluoromethyl)phenylsulfon...)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333857((R)-2-(7-(4-chloro-N-methylphenylsulfonamido)-6,7,...)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333843((R)-2-(3-chloro-2-fluoro-7-(4-fluoro-N-methylpheny...)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333853((R)-2-(7-(N,2-dimethylphenylsulfonamido)-6,7,8,9-t...)copy SMILEScopy InChI
Affinity DataKi:  51nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:Binding affinity to thromboxane receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333869((R)-2-(3-chloro-7-(4-fluoro-N-methylphenylsulfonam...)copy SMILEScopy InChI
Affinity DataKi:  104nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333865((R)-2-(7-(N-methylpyridine-2-sulfonamido)-6,7,8,9-...)copy SMILEScopy InChI
Affinity DataKi:  117nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333876((R)-2-(2,3-difluoro-7-(4-fluoro-N-methylphenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  121nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50333858((R)-2-(7-(N-methyl-4-(trifluoromethyl)phenylsulfon...)copy SMILEScopy InChI
Affinity DataKi:  123nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959HTHPubMed
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