Found 198 hits of Enzyme Inhibition Constant Data
TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 0.580nMAssay Description:Binding affinity to thromboxane receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to thromboxane receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Binding affinity to thromboxane receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 117nMAssay Description:Binding affinity to human recombinant CRTH2 receptor by cell based radioligand equilibrium competition assayMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 121nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre for Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 123nMAssay Description:Binding affinity to prostanoid DP1 receptorMore data for this Ligand-Target Pair