Compile Data Set for Download or QSAR

Found 81 hits of Enzyme Inhibition Constant Data   

TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337608(CHEMBL1683063 | cis-((1S,3R)-3-(3-ethyl-tetrahydro...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337604(CHEMBL1683059 | Cis-((1S,3R)-1-isopropyl-3-(3-meth...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Mus musculus)
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Binding affinity to mouse CCR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Rattus norvegicus)
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to rat CCR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337604(CHEMBL1683059 | Cis-((1S,3R)-1-isopropyl-3-(3-meth...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337634(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Displacement of MCP-Alexa 488 from CCR2 in human whole blood after 5 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337634(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Displacement of MCP-Alexa 488 from CCR2 in human whole blood after 5 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337608(CHEMBL1683063 | cis-((1S,3R)-3-(3-ethyl-tetrahydro...)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337619(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxytetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337612(CHEMBL1683067 | cis-((1S,3R)-1-isopropyl-3-((3S,4S...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337605(CHEMBL1683060 | Cis-((1S,3R)-1-isopropyl-3-(3-meth...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337618(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337618(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337612(CHEMBL1683067 | cis-((1S,3R)-1-isopropyl-3-((3S,4S...)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337612(CHEMBL1683067 | cis-((1S,3R)-1-isopropyl-3-((3S,4S...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Displacement of MCP-Alexa 488 from CCR2 in human whole blood after 5 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337634(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 8.40nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337620(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337634(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337622(((1S,3R)-1-ethyl-3-((3S,4S)-3-methoxy-tetrahydro-2...)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337605(CHEMBL1683060 | Cis-((1S,3R)-1-isopropyl-3-(3-meth...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337634(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human CCR5 receptor by chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337623(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337620(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337609(CHEMBL1683064 | cis-((1S,3R)-3-(3-ethyl-tetrahydro...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337633(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337613(CHEMBL1683068 | cis-((1S,3R)-1-isopropyl-3-(3-meth...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337633(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337620(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Displacement of MCP-Alexa 488 from CCR2 in human whole blood after 5 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337608(CHEMBL1683063 | cis-((1S,3R)-3-(3-ethyl-tetrahydro...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337602(((1S,3R)-1-isopropyl-3-(tetrahydro-2H-pyran-4-ylam...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337632(((1R,3R)-1-(3-fluoropropyl)-3-((3S,4S)-3-methoxy-t...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337626(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337624(((1S,3R)-1-sec-butyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337614(CHEMBL1683069 | cis-((1S,3R)-3-(3-ethoxy-tetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337612(CHEMBL1683067 | cis-((1S,3R)-1-isopropyl-3-((3S,4S...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337618(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337606(CHEMBL1683061 | trans-((1S,3R)-1-isopropyl-3-(3-me...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337625(((1R,3R)-1-(cyclopropylmethyl)-3-((3S,4S)-3-methox...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337622(((1S,3R)-1-ethyl-3-((3S,4S)-3-methoxy-tetrahydro-2...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337627(((1S,3R)-1-(ethoxymethyl)-3-((3S,4S)-3-methoxy-tet...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337620(((1S,3R)-1-isopropyl-3-((3S,4S)-3-methoxy-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Displacement of labeled MIP-1beta from human CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337616(CHEMBL1683071 | cis-((1S,3R)-1-isopropyl-3-(3-(met...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337632(((1R,3R)-1-(3-fluoropropyl)-3-((3S,4S)-3-methoxy-t...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337623(((1S,3R)-3-((3S,4S)-3-methoxy-tetrahydro-2H-pyran-...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337601(((1S,3R)-1-isopropyl-3-(tetrahydro-2H-pyran-4-ylam...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Incyte Corporation

Curated by ChEMBL
LigandPNGBDBM50337614(CHEMBL1683069 | cis-((1S,3R)-3-(3-ethoxy-tetrahydr...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6C4CPubMed
Displayed 1 to 50 (of 81 total ) | Next | Last >>* indicates data uncertainty>20%