Compile Data Set for Download or QSAR

Found 120 hits of Enzyme Inhibition Constant Data   

TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)copy SMILEScopy InChI
Affinity DataKi:  7.40nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341098((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-(3-fluor...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341104((4-(2-methoxyphenyl)piperazin-1-yl)(3-(4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341093((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-ethylphe...)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341079((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341099(2-(2-(4-(3-(4-chlorophenyl)-1H-pyrazole-5-carbonyl...)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341075((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341075((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341109((3-(2,4-dichlorophenyl)-1H-pyrazol-5-yl)(4-(2-meth...)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341105((4-(2-methoxyphenyl)piperazin-1-yl)(3-(4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50291261((S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)pip...)copy SMILEScopy InChI
Affinity DataKi:  330nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341082((5-(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)(4-(2-...)copy SMILEScopy InChI
Affinity DataKi:  350nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341081((5-(4-chlorophenyl)-1-methyl-1H-pyrazol-3-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341081((5-(4-chlorophenyl)-1-methyl-1H-pyrazol-3-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341078((S)-(3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-meth...)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341097((4-(5-chloro-2-methoxyphenyl)piperazin-1-yl)(3-(4-...)copy SMILEScopy InChI
Affinity DataKi:  400nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341076((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyb...)copy SMILEScopy InChI
Affinity DataKi:  490nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341106((4-(2-methoxyphenyl)piperazin-1-yl)(3-p-tolyl-1H-p...)copy SMILEScopy InChI
Affinity DataKi:  510nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341103((3-(4-fluorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  530nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341080((3-(4-chlorophenyl)-1-methyl-1H-pyrazol-5-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  540nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341080((3-(4-chlorophenyl)-1-methyl-1H-pyrazol-5-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  540nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341108(4-(5-(4-(2-methoxyphenyl)piperazine-1-carbonyl)-1H...)copy SMILEScopy InChI
Affinity DataKi:  700nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341074((4-(2-methoxyphenyl)piperazin-1-yl)(3-phenyl-1H-py...)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341081((5-(4-chlorophenyl)-1-methyl-1H-pyrazol-3-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341102((3-(3-fluorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341083((5-(4-chlorophenyl)isoxazol-3-yl)(4-(2-methoxyphen...)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341075((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity to human NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341076((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyb...)copy SMILEScopy InChI
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity to human NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341080((3-(4-chlorophenyl)-1-methyl-1H-pyrazol-5-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341101((3-(2-fluorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341077((3-cyclohexyl-1H-pyrazol-5-yl)(4-(2-methoxyphenyl)...)copy SMILEScopy InChI
Affinity DataKi:  2.90E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341081((5-(4-chlorophenyl)-1-methyl-1H-pyrazol-3-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341110((4-(2-methoxyphenyl)piperazin-1-yl)(3-(pyridin-2-y...)copy SMILEScopy InChI
Affinity DataKi:  3.60E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)copy SMILEScopy InChI
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341080((3-(4-chlorophenyl)-1-methyl-1H-pyrazol-5-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341076((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyb...)copy SMILEScopy InChI
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341074((4-(2-methoxyphenyl)piperazin-1-yl)(3-phenyl-1H-py...)copy SMILEScopy InChI
Affinity DataKi:  6.70E+3nMAssay Description:Binding affinity to human NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341075((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyp...)copy SMILEScopy InChI
Affinity DataKi:  8.00E+3nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341080((3-(4-chlorophenyl)-1-methyl-1H-pyrazol-5-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50051293((S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinol...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341074((4-(2-methoxyphenyl)piperazin-1-yl)(3-phenyl-1H-py...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+4nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341074((4-(2-methoxyphenyl)piperazin-1-yl)(3-phenyl-1H-py...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+4nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341081((5-(4-chlorophenyl)-1-methyl-1H-pyrazol-3-yl)(4-(2...)copy SMILEScopy InChI
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341076((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxyb...)copy SMILEScopy InChI
Affinity DataKi:  1.90E+4nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341104((4-(2-methoxyphenyl)piperazin-1-yl)(3-(4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in CHO cells assessed as inhibition of NKB-induced increase of intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341098((3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-(3-fluor...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in CHO cells assessed as inhibition of NKB-induced increase of intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
Displayed 1 to 50 (of 120 total ) | Next | Last >>* indicates data uncertainty>20%