Found 120 hits of Enzyme Inhibition Constant Data
Affinity DataKi: 1.90nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to human NK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity to human NK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.60E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.70E+3nMAssay Description:Binding affinity to human NK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human NK1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity to human NK2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in CHO cells assessed as inhibition of NKB-induced increase of intracellular calcium ...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in CHO cells assessed as inhibition of NKB-induced increase of intracellular calcium ...More data for this Ligand-Target Pair