Found 139 hits of Enzyme Inhibition Constant Data
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetRibosomal protein S6 kinase alpha-5(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of MSK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 3(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of MST2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of PRK2More data for this Ligand-Target Pair
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of TIE2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of IDO1More data for this Ligand-Target Pair
TargetEphrin type-B receptor 2(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of EPHB2More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of TBK1More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of AURORA AMore data for this Ligand-Target Pair
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of CAMK1DMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of DYRK1AMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of Itk after 40 mins by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of Itk after 40 mins by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of ERK1More data for this Ligand-Target Pair
TargetProtein kinase C theta type(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of Itk after 40 mins by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of ZAP70More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of ERK2More data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of C-RAFMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of Itk after 40 mins by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of Itk after 40 mins by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of Itk after 40 mins by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of Itk after 40 mins by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair