Compile Data Set for Download or QSAR

Found 61 hits of Enzyme Inhibition Constant Data   

TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353042(CHEMBL1822521)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353041(CHEMBL1822520)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353039(CHEMBL1821735)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353048(CHEMBL1822527)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353044(CHEMBL1822523)copy SMILEScopy InChI
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353043(CHEMBL1822522)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353045(CHEMBL1822524)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353040(CHEMBL1822519)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353046(CHEMBL1822525)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353047(CHEMBL1822526)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353051(CHEMBL1822514)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353052(CHEMBL1822515)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353056(CHEMBL1822513)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353051(CHEMBL1822514)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353056(CHEMBL1822513)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353048(CHEMBL1822527)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353046(CHEMBL1822525)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353044(CHEMBL1822523)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353047(CHEMBL1822526)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353042(CHEMBL1822521)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353043(CHEMBL1822522)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353040(CHEMBL1822519)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353041(CHEMBL1822520)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353052(CHEMBL1822515)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353042(CHEMBL1822521)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353050(CHEMBL1822512)copy SMILEScopy InChI
Affinity DataIC50: 194nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353045(CHEMBL1822524)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of NPM/ALK phosphorylation in human KARPAS299 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353041(CHEMBL1822520)copy SMILEScopy InChI
Affinity DataIC50: 206nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353049(CHEMBL1822511)copy SMILEScopy InChI
Affinity DataIC50: 212nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353055(CHEMBL1822518)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353044(CHEMBL1822523)copy SMILEScopy InChI
Affinity DataIC50: 266nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353049(CHEMBL1822511)copy SMILEScopy InChI
Affinity DataIC50: 295nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353053(CHEMBL1822516)copy SMILEScopy InChI
Affinity DataIC50: 326nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353043(CHEMBL1822522)copy SMILEScopy InChI
Affinity DataIC50: 357nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353039(CHEMBL1821735)copy SMILEScopy InChI
Affinity DataIC50: 366nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353040(CHEMBL1822519)copy SMILEScopy InChI
Affinity DataIC50: 391nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353053(CHEMBL1822516)copy SMILEScopy InChI
Affinity DataIC50: 726nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353048(CHEMBL1822527)copy SMILEScopy InChI
Affinity DataIC50: 809nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353054(CHEMBL1822517)copy SMILEScopy InChI
Affinity DataIC50: 883nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353045(CHEMBL1822524)copy SMILEScopy InChI
Affinity DataIC50: 934nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353046(CHEMBL1822525)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353047(CHEMBL1822526)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353055(CHEMBL1822518)copy SMILEScopy InChI
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353050(CHEMBL1822512)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant ALK assessed as phosphorylated product using PLC-gamma/GST substrate by modified ELISA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetInsulin receptor(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353054(CHEMBL1822517)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353046(CHEMBL1822525)copy SMILEScopy InChI
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human ERG channel by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353052(CHEMBL1822515)copy SMILEScopy InChI
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353046(CHEMBL1822525)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353046(CHEMBL1822525)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Cephalon, Inc.

Curated by ChEMBL
LigandPNGBDBM50353046(CHEMBL1822525)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP1A2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ331FPubMed
Displayed 1 to 50 (of 61 total ) | Next | Last >>* indicates data uncertainty>20%