Compile Data Set for Download or QSAR

Found 52 hits of Enzyme Inhibition Constant Data   

TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419188(CHEMBL1616460)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419176(CHEMBL1831027)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419186(CHEMBL1545942)copy SMILEScopy InChI
Affinity DataKi:  398nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419198(CHEMBL1828843)copy SMILEScopy InChI
Affinity DataKi:  398nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419190(CHEMBL1828844)copy SMILEScopy InChI
Affinity DataKi:  501nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419180(CHEMBL1831037)copy SMILEScopy InChI
Affinity DataKi:  501nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419192(CHEMBL1828846)copy SMILEScopy InChI
Affinity DataKi:  631nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419178(CHEMBL1831029)copy SMILEScopy InChI
Affinity DataKi:  631nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419175(CHEMBL1831034)copy SMILEScopy InChI
Affinity DataKi:  794nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419185(CHEMBL1831048)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353946(CHEMBL1831032)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM74511(1-(1-benzothien-3-ylmethyl)piperidine | 1-(1-benzo...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419177(CHEMBL1831028)copy SMILEScopy InChI
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419200(CHEMBL1740345)copy SMILEScopy InChI
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419189(CHEMBL1619901)copy SMILEScopy InChI
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419191(CHEMBL1828845)copy SMILEScopy InChI
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419187(CHEMBL1624521)copy SMILEScopy InChI
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419197(CHEMBL1831047)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353944(CHEMBL1831036)copy SMILEScopy InChI
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419194(CHEMBL1828849)copy SMILEScopy InChI
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419195(CHEMBL1828847)copy SMILEScopy InChI
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419191(CHEMBL1828845)copy SMILEScopy InChI
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419181(CHEMBL1831042)copy SMILEScopy InChI
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419182(CHEMBL1831044)copy SMILEScopy InChI
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;bromide | 2-acet...)copy SMILEScopy InChI
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;bromide | 2-acet...)copy SMILEScopy InChI
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419180(CHEMBL1831037)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353947(CHEMBL1831030)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419184(CHEMBL1831046)copy SMILEScopy InChI
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419179(CHEMBL1831035)copy SMILEScopy InChI
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419183(CHEMBL1831045)copy SMILEScopy InChI
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353945(CHEMBL1831033)copy SMILEScopy InChI
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419199(CHEMBL1828848)copy SMILEScopy InChI
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419188(CHEMBL1616460)copy SMILEScopy InChI
Affinity DataKi:  1.58E+4nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM74511(1-(1-benzothien-3-ylmethyl)piperidine | 1-(1-benzo...)copy SMILEScopy InChI
Affinity DataKi:  1.58E+4nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419185(CHEMBL1831048)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419187(CHEMBL1624521)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419176(CHEMBL1831027)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Displacement of [3H]-MLA from human alpha7 nAChR expressed in human SH-SY5Y cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419196(CHEMBL1831040)copy SMILEScopy InChI
Affinity DataKi:  2.51E+4nMAssay Description:Displacement of [3H]-epibatidine from histidine-tagged Lymnaea stagnalis AChBP expressed in Sf9 cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419181(CHEMBL1831042)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419182(CHEMBL1831044)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419175(CHEMBL1831034)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353946(CHEMBL1831032)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50419179(CHEMBL1831035)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353945(CHEMBL1831033)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353948(CHEMBL1831043)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353947(CHEMBL1831030)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
VU University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50353949(CHEMBL1831038)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus oocytes assessed as increase of acetylcholine-induced effect by electrophysiology assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN09BHPubMed
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